messages
listlengths
2
10
metadata
dict
[ { "role": "user", "content": "What drugs target Endothelin receptor type B? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Endothelin receptor type B\n\nThe following approved drugs are known to interact with En...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Zone of skin? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Zone of skin\n\nThe following approved drugs are known to interact with Zone of skin:\n\n - **BARBITA...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target D(4) dopamine receptor? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting D(4) dopamine receptor\n\nThe following approved drugs are known to interact with D(4) dopam...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Sigma non-opioid intracellular receptor 1? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Sigma non-opioid intracellular receptor 1\n\nThe following approved drugs...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Phospholipidosis? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Phospholipidosis\n\nThe following approved drugs are known to interact with Phospholipidosis:\n\n ...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Trypanothione reductase? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Trypanothione reductase\n\nThe following approved drugs are known to interact with Trypanot...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Glutathione reductase, mitochondrial? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Glutathione reductase, mitochondrial\n\nThe following approved drugs are known...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Prothrombin? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Prothrombin\n\nThe following approved drugs are known to interact with Prothrombin:\n\n - **MELAGATRAN...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Translocator protein? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Translocator protein\n\nThe following approved drugs are known to interact with Translocator p...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Survival motor neuron protein? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Survival motor neuron protein\n\nThe following approved drugs are known to interact w...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Prelamin-A/C? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Prelamin-A/C\n\nThe following approved drugs are known to interact with Prelamin-A/C:\n\n - **SULFAME...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Pasteurella multocida? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Pasteurella multocida\n\nThe following approved drugs are known to interact with Pasteurella ...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target P388? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting P388\n\nThe following approved drugs are known to interact with P388:\n\n - **AMSACRINE** (ChEMBL: CHEMBL43):...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target L1210? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting L1210\n\nThe following approved drugs are known to interact with L1210:\n\n - **AMSACRINE** (ChEMBL: CHEMBL4...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target DNA topoisomerase II? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting DNA topoisomerase II\n\nThe following approved drugs are known to interact with DNA topoisomer...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Felis catus? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Felis catus\n\nThe following approved drugs are known to interact with Felis catus:\n\n - **ETHACRYNIC...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Chymotrypsin-C? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Chymotrypsin-C\n\nThe following approved drugs are known to interact with Chymotrypsin-C:\n\n - **G...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Cricetinae gen. sp.? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Cricetinae gen. sp.\n\nThe following approved drugs are known to interact with Cricetinae gen. ...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Melatonin receptor type 1B? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Melatonin receptor type 1B\n\nThe following approved drugs are known to interact with Me...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Melatonin receptor? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Melatonin receptor\n\nThe following approved drugs are known to interact with Melatonin receptor...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Melatonin receptor type 1A? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Melatonin receptor type 1A\n\nThe following approved drugs are known to interact with Me...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Serotonin 2 (5-HT2) receptor? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Serotonin 2 (5-HT2) receptor\n\nThe following approved drugs are known to interact wit...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target 5-hydroxytryptamine receptor 2A? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting 5-hydroxytryptamine receptor 2A\n\nThe following approved drugs are known to intera...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Adrenergic receptor alpha-1? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Adrenergic receptor alpha-1\n\nThe following approved drugs are known to interact with ...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Histamine H1 receptor? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Histamine H1 receptor\n\nThe following approved drugs are known to interact with Histamine H1...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target 5-hydroxytryptamine receptor 1B? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting 5-hydroxytryptamine receptor 1B\n\nThe following approved drugs are known to intera...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target D(1A) dopamine receptor? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting D(1A) dopamine receptor\n\nThe following approved drugs are known to interact with D(1A) do...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Adrenergic receptor alpha? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Adrenergic receptor alpha\n\nThe following approved drugs are known to interact with Adre...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Trypanosoma brucei? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Trypanosoma brucei\n\nThe following approved drugs are known to interact with Trypanosoma brucei...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target ATP-binding cassette sub-family C member 2? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting ATP-binding cassette sub-family C member 2\n\nThe following approved dru...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Cellular retinoic acid-binding protein 1? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Cellular retinoic acid-binding protein 1\n\nThe following approved drugs a...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Human immunodeficiency virus 1? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Human immunodeficiency virus 1\n\nThe following approved drugs are known to interact...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target MT4? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting MT4\n\nThe following approved drugs are known to interact with MT4:\n\n - **NEVIRAPINE** (ChEMBL: CHEMBL57): S...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Human immunodeficiency virus type 1 reverse transcriptase? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Human immunodeficiency virus type 1 reverse transcriptase...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target HT-29? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting HT-29\n\nThe following approved drugs are known to interact with HT-29:\n\n - **MITOXANTRONE** (ChEMBL: CHEM...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target B16? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting B16\n\nThe following approved drugs are known to interact with B16:\n\n - **MITOXANTRONE** (ChEMBL: CHEMBL58):...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Human immunodeficiency virus type 1 integrase? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Human immunodeficiency virus type 1 integrase\n\nThe following approv...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Tubulin? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Tubulin\n\nThe following approved drugs are known to interact with Tubulin:\n\n - **PODOFILOX** (ChEMBL: C...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Tetrahymena pyriformis? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Tetrahymena pyriformis\n\nThe following approved drugs are known to interact with Tetrahymen...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target KB? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting KB\n\nThe following approved drugs are known to interact with KB:\n\n - **PODOFILOX** (ChEMBL: CHEMBL61): SMILE...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Mycobacterium avium? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Mycobacterium avium\n\nThe following approved drugs are known to interact with Mycobacterium av...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Vero? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Vero\n\nThe following approved drugs are known to interact with Vero:\n\n - **ISONIAZID** (ChEMBL: CHEMBL64):...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target PBMC? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting PBMC\n\nThe following approved drugs are known to interact with PBMC:\n\n - **THALIDOMIDE** (ChEMBL: CHEMBL46...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target CCRF-CEM? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting CCRF-CEM\n\nThe following approved drugs are known to interact with CCRF-CEM:\n\n - **ADENOSINE** (ChEMBL...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Adenosine receptor A1? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Adenosine receptor A1\n\nThe following approved drugs are known to interact with Adenosine re...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Opioid receptors; mu/kappa/delta? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Opioid receptors; mu/kappa/delta\n\nThe following approved drugs are known to inte...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Mu-type opioid receptor? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Mu-type opioid receptor\n\nThe following approved drugs are known to interact with Mu-type ...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Opioid receptor? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Opioid receptor\n\nThe following approved drugs are known to interact with Opioid receptor:\n\n - ...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "What drugs target Monkey? Compare their molecular structures and discuss their mechanism of action." }, { "role": "assistant", "content": "## Drugs Targeting Monkey\n\nThe following approved drugs are known to interact with Monkey:\n\n - **CODEINE** (ChEMBL: CHEMBL...
{ "pillar": "discovery", "domain": "drug-target interaction", "skill_type": "requires-knowledge", "source": "chembl", "difficulty": "intermediate" }
[ { "role": "user", "content": "Given that CHEMBL324340 shows IC50 of 2500.0 nM against Heparanase, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 2500.0 nM against Heparan...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL109600 shows IC50 of 9000.0 nM against Heparanase, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 9000.0 nM against Heparan...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL357278 shows IC50 of 4000.0 nM against Peroxisomal acyl-coenzyme A oxidase 1, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 ...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL357119 shows IC50 of 17000.0 nM against Peroxisomal acyl-coenzyme A oxidase 1, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL152968 shows IC50 of 180.0 nM against Peroxisomal acyl-coenzyme A oxidase 1, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 =...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL152968 shows IC50 of 6000.0 nM against Cytochrome P450 1A2, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 6000.0 nM agains...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL152968 shows IC50 of 37000.0 nM against Cytochrome P450 3A4, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 37000.0 nM agai...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL152968 shows IC50 of 24000.0 nM against Cytochrome P450 2C9, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 24000.0 nM agai...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268177 shows Ki of 6000.0 nM against Carbonic anhydrase 1, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 6000.0 nM against C...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268177 shows Ki of 70.0 nM against Carbonic anhydrase 2, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 70.0 nM against Carbo...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268177 shows Ki of 285.0 nM against Carbonic anhydrase 9, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 285.0 nM against Car...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268177 shows Ki of 50.0 nM against Carbonic anhydrase 13, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 50.0 nM against Carb...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268439 shows Ki of 6.0 nM against Carbonic anhydrase 1, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 6.0 nM against Carboni...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268439 shows Ki of 2.0 nM against Carbonic anhydrase 2, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 2.0 nM against Carboni...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268439 shows Ki of 38.0 nM against Carbonic anhydrase 9, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 38.0 nM against Carbo...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL268439 shows Ki of 2.0 nM against Carbonic anhydrase 13, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 2.0 nM against Carbon...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL54530 shows Ki of 19010.78 nM against DNA topoisomerase 3, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 19010.78 nM against...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL54530 shows Ki of 158124.8 nM against DNA topoisomerase 3, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 158124.8 nM against...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL302907 shows Kd of 25.12 nM against Histamine H2 receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 25.12 nM against Hi...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL302907 shows Kd of 125892.54 nM against Histamine H1 receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 125892.54 nM ag...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL302907 shows Kd of 398107.17 nM against Unchecked, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 398107.17 nM against Unchec...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL302907 shows Kd of 50118.72 nM against Adrenergic receptor beta, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 50118.72 nM a...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL429345 shows IC50 of 0.009 ug.mL-1 against Enterococcus faecium, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 0.009 ug.mL...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL429345 shows IC50 of 0.056 ug.mL-1 against Lacticaseibacillus casei, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 0.056 u...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL429345 shows IC50 of 0.064 ug.mL-1 against Lacticaseibacillus casei, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 0.064 u...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL415997 shows IC50 of 2.9 ug.mL-1 against Cavia porcellus, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 2.9 ug.mL-1 agains...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL13299 shows Kd of 7.943 nM against Cavia porcellus, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 7.943 nM against Cavia por...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL13299 shows Kd of 199.53 nM against Cavia porcellus, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 199.53 nM against Cavia p...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL305153 shows Kd of 37.15 nM against Beta-1 adrenergic receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 37.15 nM again...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL305153 shows Kd of 16.98 nM against Beta-2 adrenergic receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 16.98 nM again...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL305153 shows IC50 of 29.4 nM against Beta-1 adrenergic receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 29.4 nM aga...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL305153 shows IC50 of 30.8 nM against Beta-2 adrenergic receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 30.8 nM aga...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL156707 shows IC50 of 1584.89 nM against Malate dehydrogenase, mitochondrial, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 =...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL13228 shows Kd of 0.3981 nM against Cavia porcellus, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 0.3981 nM against Cavia p...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL13228 shows Kd of 0.7943 nM against Cavia porcellus, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 0.7943 nM against Cavia p...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL279087 shows IC50 of 120.0 nM against GABA-A receptor; anion channel, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 120.0 ...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL279969 shows IC50 of 1850.0 nM against GABA-A receptor; anion channel, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 1850....
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL20214 shows IC50 of 34.0 nM against GABA-A receptor; anion channel, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 34.0 nM ...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL277617 shows IC50 of 107.0 nM against GABA-A receptor; anion channel, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 107.0 ...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL408689 shows Kd of 5011.87 nM against Rattus norvegicus, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Kd = 5011.87 nM against Ra...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL3350133 shows IC50 of 22.0 nM against Opioid receptors; mu & kappa, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 22.0 nM ...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL3350133 shows Ki of 44.0 nM against Mu-type opioid receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 44.0 nM against M...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL3350133 shows Ki of 590.0 nM against Kappa-type opioid receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 590.0 nM agai...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL3350133 shows Ki of 110.0 nM against Delta-type opioid receptor, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 110.0 nM agai...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL15886 shows IC50 of 100000.0 nM against Acetylcholinesterase, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 100000.0 nM ag...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL15886 shows IC50 of 170000.0 nM against Acetylcholinesterase, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 170000.0 nM ag...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL63484 shows Ki of 1400000.0 nM against Pancreatic elastase, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 1400000.0 nM again...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL294543 shows Ki of 2410000.0 nM against Pancreatic elastase, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of Ki = 2410000.0 nM agai...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL1202755 shows IC50 of 8000.0 nM against Cavia porcellus, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 8000.0 nM against C...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL1202755 shows IC50 of 1000.0 nM against Thromboxane-A synthase, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 1000.0 nM ag...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }
[ { "role": "user", "content": "Given that CHEMBL542565 shows IC50 of 870.0 nM against L1210, what does this suggest about its potential as a drug candidate? Discuss selectivity and potency considerations." }, { "role": "assistant", "content": "## Analysis of IC50 = 870.0 nM against L1210\n\n### P...
{ "pillar": "discovery", "domain": "ADMET", "skill_type": "requires-reasoning", "source": "chembl", "difficulty": "advanced" }